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Kinase Inhibitors

Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells.

Why are kinase inhibitors prescribed?

How are these percentages calculated?

Key takeaways

Kinase inhibitors are a broad group of medications used to treat several types of cancer, such as lung cancer, breast cancer, and leukemia. They also have other uses, such as treating graft-versus-host disease. These medications work by blocking specific enzymes called kinases, which help stop the growth and spread of cancer cells (or inflammatory cells). Kinase inhibitors often come as oral pills. Examples include Gleevec (imatinib), Tykerb (lapatinib), Rezurock (belumosudil), and more.

Prices for popular Kinase Inhibitors medications

Viewing 25 of 83 medications

Gleevec (imatinib)

as low as$100

IMATINIB treats some types of cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Rhopressa

as low as$335

Rhopressa (Netarsudil) is used to treat open-angle glaucoma and high pressure in the eye. There is currently no generic alternative to Rhopressa. The most common version of Rhopressa is covered by 73% of insurance plans at a co-pay of $60.00-$80.00, however, some pharmacy coupons or cash prices may be lower.

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Imkeldi

as low as$2,322

Imkeldi is part of the Kinase Inhibitors class and treats Mastocytosis, Skin Cancer, GIST and other conditions. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Imkeldi is only available as a brand name drug.

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Tasigna (nilotinib)

as low as$3,018

NILOTINIB treats leukemia. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Rhapsido

as low as$4,331

Rhapsido is part of the Kinase Inhibitors class and treats Hives. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Rhapsido is only available as a brand name drug.

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Danziten

as low as$4,625

Danziten is part of the Kinase Inhibitors class and treats Leukemia. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Danziten is only available as a brand name drug.

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Augtyro

as low as$7,651

REPOTRECTINIB treats lung cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Ensacove

as low as$8,916

Ensacove is part of the Kinase Inhibitors class and treats Lung Cancer. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Ensacove is only available as a brand name drug.

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Tepmetko

as low as$12,637

TEPOTINIB treats lung cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Lazcluze

as low as$17,421

Lazcluze is part of the Kinase Inhibitors class and treats Lung Cancer. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Lazcluze is only available as a brand name drug.

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Votrient (pazopanib)

as low as$17,560

PAZOPANIB treats kidney cancer. It may also be used to treat sarcoma, a cancer that occurs in bone and connective tissues, such as fat, muscle, and blood vessels. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Vanflyta

as low as$17,654

QUIZARTINIB treats leukemia. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Afinitor Disperz

as low as$18,857

View othermTOR Inhibitors

EVEROLIMUS treats some types of cancer. It may also be used to treat symptoms of tuberous sclerosis, a genetic condition that causes benign tumors to grow in the brain and other parts of the body. It works by slowing or stopping the growth of tumor cells.

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Fruzaqla

as low as$19,288

FRUQUINTINIB treats colorectal cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Truseltiq

as low as$21,598

INFIGRATINIB treats bile duct cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Joenja

as low as$24,388

LENIOLISIB treats activated phosphoinositide 3-kinase delta syndrome (APDS). It works by balancing substances in your body that help regulate the immune system. This helps your body make mature white blood cells, which protect your body from infection.

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Vonjo

as low as$24,760

PACRITINIB treats bone marrow cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Turalio

as low as$24,923

PEXIDARTINIB treats noncancerous tumors that occur in joints. It works by blocking a protein that causes tumor cells to grow and multiply.

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Vijoice

as low as$31,090

ALPELISIB treats symptoms of PIK3CA-related overgrowth spectrum (PROS), a group of conditions that cause extra tissue growth in different parts of the body. It works by blocking a protein that causes cells to grow and multiply. This helps to slow tissue growth.

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Ojemda

as low as$37,023

Ojemda is part of the Kinase Inhibitors class and treats Brain Tumor. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Ojemda is only available as a brand name drug.

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Alecensa

ALECTINIB treats lung cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Aliqopa

COPANLISIB treats lymphoma. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

Alunbrig

BRIGATINIB treats lung cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Avmapki Fakzynja Co-Pack

Avmapki Fakzynja Co-Pack is part of the Kinase Inhibitors class and treats Ovarian Cancer. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Avmapki Fakzynja Co-Pack is only available as a brand name drug.

Ayvakit

The average list price of Ayvakit (Avapritinib) is $38,929.00, but your out of pocket cost will likely be less if you have insurance. Ayvakit is covered by some Medicare and insurance plans. This drug is also a limited distribution drug, meaning it is not available at retail pharmacies. Refer to the Key Takeaways for additional information on Ayvakit and check our savings tips for other ways to reduce your cost. A generic version of Ayvakit is not yet available.

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Disclaimer: Popularity is based on total prescriptions for the brand and generic versions of each drug, regardless of the condition being treated. Some drugs are prescribed for multiple conditions.

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