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Kinase Inhibitors

Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells.

Why are kinase inhibitors prescribed?

How are these percentages calculated?

Key takeaways

Kinase inhibitors are a broad group of medications used to treat several types of cancer, such as lung cancer, breast cancer, and leukemia. They also have other uses, such as treating graft-versus-host disease. These medications work by blocking specific enzymes called kinases, which help stop the growth and spread of cancer cells (or inflammatory cells). Kinase inhibitors often come as oral pills. Examples include Gleevec (imatinib), Tykerb (lapatinib), Rezurock (belumosudil), and more.

Prices for popular Kinase Inhibitors medications

Viewing 25 of 38 medications

Truqap

CAPIVASERTIB treats breast cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Ibtrozi

Ibtrozi is part of the Kinase Inhibitors class and treats Lung Cancer. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Ibtrozi is only available as a brand name drug.

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Ofev (Nintedanib)

Ofev is part of the Kinase Inhibitors class and treats Idiopathic Pulmonary Fibrosis. Ofev is only available as a brand name drug.

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Lorbrena

LORLATINIB treats lung cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Romvimza

Romvimza is part of the Kinase Inhibitors class and treats Giant Cell Tumor. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Romvimza is only available as a brand name drug.

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Sutent (Sunitinib)

Sutent (Sunitinib) is an expensive drug that targets proteins in cancer cells and stops the cancer cells from growing. It is used to treat specific digestive tract tumors called GISTs, advanced kidney cancer, and certain pancreatic neuroendocrine tumors. It is less popular than comparable drugs. While 99% of insurance plans cover the most common version of Sutent at a co-pay of $32.50-$60.00, many of them have restrictions.

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Dasatinib

as low as$737

Dasatinib is part of the Kinase Inhibitors class and treats Leukemia. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Dasatinib is only available as a generic drug.

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Ensacove

as low as$2,511

Ensacove is only available as a brand name drug.

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Nilotinib

as low as$5,352

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Votrient (Pazopanib)

as low as$9,403

PAZOPANIB treats kidney cancer. It may also be used to treat sarcoma, a cancer that occurs in bone and connective tissues, such as fat, muscle, and blood vessels. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Turalio

as low as$13,292

PEXIDARTINIB treats noncancerous tumors that occur in joints. It works by blocking a protein that causes tumor cells to grow and multiply.

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Vonjo

as low as$27,376

PACRITINIB treats bone marrow cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Augtyro

as low as$32,734

REPOTRECTINIB treats lung cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Jideytro

as low as$34,513

Jideytro is part of the Kinase Inhibitors class and treats Lung Cancer. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Jideytro is only available as a brand name drug.

Atebrioz

as low as$34,875

Atebrioz is part of the Kinase Inhibitors class and treats Connective Tissue Disorders. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Atebrioz is only available as a brand name drug.

Lisraya

as low as$35,836

Lisraya is part of the Kinase Inhibitors class and treats Dermatomyositis. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Lisraya is only available as a brand name drug.

Ojemda

as low as$42,399

Ojemda is part of the Kinase Inhibitors class and treats Brain Tumor. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Ojemda is only available as a brand name drug.

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Revtorpyk

Revtorpyk is part of the Kinase Inhibitors class and treats Breast Cancer. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Revtorpyk is only available as a brand name drug.

Rydapt

MIDOSTAURIN treats blood and bone marrow cancers. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Tavalisse

FOSTAMATINIB treats low levels of platelets in your body caused by immune thrombocytopenia (ITP). It is prescribed when other medications have not worked well enough. It works by increasing the amount of platelets in your blood. This lowers the risk of bleeding.

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Subject to eligibility

Lenvima

as low as$0

LENVATINIB treats some types of cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Alecensa

ALECTINIB treats lung cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Alunbrig

BRIGATINIB treats lung cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.

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Avmapki Fakzynja Co-Pack

Avmapki Fakzynja Co-Pack is part of the Kinase Inhibitors class and treats Ovarian Cancer. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Avmapki Fakzynja Co-Pack is only available as a brand name drug.

Ayvakit

The average list price of Ayvakit (Avapritinib) is $38,929.00, but your out of pocket cost will likely be less if you have insurance. Ayvakit is covered by some Medicare and insurance plans. This drug is also a limited distribution drug, meaning it is not available at retail pharmacies. Refer to the Key Takeaways for additional information on Ayvakit and check our savings tips for other ways to reduce your cost. A generic version of Ayvakit is not yet available.

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Disclaimer: Popularity is based on total prescriptions for the brand and generic versions of each drug, regardless of the condition being treated. Some drugs are prescribed for multiple conditions.

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