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Kinase Inhibitors

Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells.

Why are kinase inhibitors prescribed?

  1. Leukemia (15%)
  2. GIST (14%)
  3. Soft Tissue Sarcoma (14%)
  4. Mastocytosis (14%)
  5. Myelodysplastic Syndromes (14%)
  6. Glaucoma (12%)
  7. Eye Pressure (12%)
  8. Lung Cancer (0%)
  9. Melanoma (0%)
  10. Renal Cancer (0%)

Key takeaways

Kinase inhibitors are a broad group of medications used to treat several types of cancer, such as lung cancer, breast cancer, and leukemia. They also have other uses, such as treating graft-versus-host disease. These medications work by blocking specific enzymes called kinases, which help stop the growth and spread of cancer cells (or inflammatory cells). Kinase inhibitors often come as oral pills. Examples include Gleevec (imatinib), Tykerb (lapatinib), Rezurock (belumosudil), and more.

Prices for popular Kinase Inhibitors medications
Viewing 25 of 85 medications
IMATINIB treats some types of cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.
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Rhopressa

as low as$326
Rhopressa (Netarsudil) is used to treat open-angle glaucoma and high pressure in the eye. There is currently no generic alternative to Rhopressa. The most common version of Rhopressa is covered by 73% of insurance plans at a co-pay of $60.00-$80.00, however, some pharmacy coupons or cash prices may be lower.
LAPATINIB treats breast cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.
Sutent (Sunitinib) is an expensive drug that targets proteins in cancer cells and stops the cancer cells from growing. It is used to treat specific digestive tract tumors called GISTs, advanced kidney cancer, and certain pancreatic neuroendocrine tumors. It is less popular than comparable drugs. While 99% of insurance plans cover the most common version of Sutent at a co-pay of $32.50-$60.00, many of them have restrictions.
DASATINIB treats leukemia. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.
Torisel (Temsirolimus) is an expensive drug that alters immune system response in the body. It is used to treat renal cell cancer.It is less popular than comparable drugs. It is available in brand and generic form. The most common version of Torisel is covered by 97% of insurance plans at a co-pay of $45.00-$73.75.
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Cosela

as low as$1,551
TRILACICLIB prevents low levels of red blood cells, white blood cells, and platelets caused by chemotherapy. It works by protecting the cells in your bone marrow that make these blood cells. This lowers the risk of infection and bleeding. It also reduces the need for blood transfusions.
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Imkeldi

as low as$2,378
Imkeldi is only available as a brand name drug.
NILOTINIB treats leukemia. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.
SORAFENIB treats some types of cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.
Rhapsido is part of the Kinase Inhibitors class and treats Hives. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Rhapsido is only available as a brand name drug.
Danziten is only available as a brand name drug.
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Augtyro

as low as$4,910
REPOTRECTINIB treats lung cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.
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Aliqopa

as low as$5,035
COPANLISIB treats lymphoma. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.
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Lytgobi

as low as$5,197
FUTIBATINIB treats bile duct cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.
PIRTOBRUTINIB treats leukemia and lymphoma. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.
Ensacove is part of the Kinase Inhibitors class and treats Lung Cancer. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Ensacove is only available as a brand name drug.
FRUQUINTINIB treats colorectal cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.
ERDAFITINIB treats bladder cancer and kidney cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.
Itovebi is part of the Kinase Inhibitors class and treats Breast Cancer. Kinase inhibitors are used to treat cancers such as leukemia, breast cancer, melanoma, lung cancer, and renal cancer. They are also used to prevent organ transplant rejection. They work by stopping cancer cell growth and preventing the spread of the cells. Itovebi is only available as a brand name drug.
TEPOTINIB treats lung cancer. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.
QUIZARTINIB treats leukemia. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.
PAZOPANIB treats kidney cancer. It may also be used to treat sarcoma, a cancer that occurs in bone and connective tissues, such as fat, muscle, and blood vessels. It works by blocking a protein that causes cancer cells to grow and multiply. This helps to slow or stop the spread of cancer cells.
Lazcluze is only available as a brand name drug.
Phyrago is only available as a brand name drug.
Disclaimer: Popularity is based on total prescriptions for the brand and generic versions of each drug, regardless of the condition being treated. Some drugs are prescribed for multiple conditions.

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